DISCOVERY OF A NOVEL CLASS OF TRIAZOLONES AS CHECKPOINT KINASE INHIBITORS - HIT TO LEAD EXPLORATION

PDB Details

PDB ID
2X8I
Status
CURRENT
Deposition Date
2010-03-09
Modification Date
2010-08-25
Pubmed ID
20673630
Method
X-RAY DIFFRACTION
Resolution (Å)
1.92
UniProt Accessions
O14757

Mapping Results

Chain Terminus Site Consensus Site Rank Consensus Site Population
A C CMP 3 15
A C EDI 4 14
A C PDIG 6 7
A N ATP 0 24
A N MPP 1 16
A N MPP 2 14
A N MT3 3 14
A N MT3 4 10
A N MT3 5 5

Mapping Results Viewer

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Legend

Color Name Hit Count