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6-Amino-4-(pyrimidin-4-yl)pyridones: Novel Glycogen Synthase Kinase-3 Inhibitors
PDB Details
PDB ID
3Q3B
Status
CURRENT
Deposition Date
2010-12-21
Modification Date
2011-06-15
Pubmed ID
21295469
Method
X-RAY DIFFRACTION
Resolution (Å)
2.7
UniProt Accessions
P49841
Mapping Results
Chain
Terminus
Site
Consensus Site Rank
Consensus Site Population
A
C
DRS
1
15
A
C
EDI
2
13
A
C
DRS
4
9
A
C
PDIG
7
5
A
N
DFG
4
8
A
N
ATP
6
6
B
C
EDI
1
13
B
C
DRS
3
11
B
C
PDIG
5
8
B
C
DRS
6
7
B
N
ATP
1
16
B
N
MT3
5
13
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Chain: B
Chain: A
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Color
Name
Hit Count
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Chain: B
Chain: A