Discovery of a Novel, Potent and Selective Inhibitor of 3-Phosphoinositide Dependent Kinase (PDK1)

PDB Details

PDB ID
3RWQ
Status
CURRENT
Deposition Date
2011-05-09
Modification Date
2011-12-28
Pubmed ID
22040023
Method
X-RAY DIFFRACTION
Resolution (Å)
2.55
UniProt Accessions
O15530

Mapping Results

Chain Terminus Site Consensus Site Rank Consensus Site Population
A C AAS 1 19
A C DRS 3 15
A C DRS 5 10
A N PIF 0 18
A N ATP 4 10
A N ATP 6 6
A N PIF 7 5
A N ATP 8 3

Mapping Results Viewer

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Legend

Color Name Hit Count