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Identification of 2-(4-pyridyl)thienopyridinones as GSK-3beta inhibitors
PDB Details
PDB ID
3ZRL
Status
CURRENT
Deposition Date
2011-06-17
Modification Date
2012-04-25
Pubmed ID
21764580
Method
X-RAY DIFFRACTION
Resolution (Å)
2.48
UniProt Accessions
P49841
Mapping Results
Chain
Terminus
Site
Consensus Site Rank
Consensus Site Population
A
C
EDI
1
17
A
C
DRS
2
16
A
C
PMP
4
6
A
C
PDIG
7
3
A
C
EDI
9
2
A
N
ATP
2
16
A
N
MT3
6
3
B
C
EDI
2
17
B
C
PDIG
5
5
B
C
DRS
8
2
B
N
ATP
1
17
B
N
MT3
6
3
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Chain: A
Chain: B
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Name
Hit Count
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Chain: A
Chain: B