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Structure of PIM-1 kinase bound to N-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
PDB Details
PDB ID
4K0Y
Status
CURRENT
Deposition Date
2013-04-04
Modification Date
2013-05-22
Pubmed ID
23623490
Method
X-RAY DIFFRACTION
Resolution (Å)
1.95
UniProt Accessions
P11309
Mapping Results
Chain
Terminus
Site
Consensus Site Rank
Consensus Site Population
A
C
EDI
2
16
A
C
DRS
3
14
A
C
CMP
5
8
A
C
PDIG
6
5
A
C
LBP
7
2
A
C
DRS
8
2
A
N
ATP
0
16
A
N
DFG
3
12
A
N
MT3
6
8
A
N
ATP
7
3
A
N
ATP
8
3
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Chain: A
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Name
Hit Count
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Chain: A