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Crystal structure of human Pim-1 kinase in complex with a quinazolinone-pyrrolopyrrolone inhibitor.
PDB Details
PDB ID
5IPJ
Status
CURRENT
Deposition Date
2016-03-09
Modification Date
2016-07-27
Pubmed ID
27285051
Method
X-RAY DIFFRACTION
Resolution (Å)
2.1
UniProt Accessions
P11309
Mapping Results
Chain
Terminus
Site
Consensus Site Rank
Consensus Site Population
A
C
EDI
2
16
A
C
DRS
3
15
A
C
DRS
5
6
A
C
PDIG
6
4
A
C
CMP
8
3
A
N
ATP
1
17
A
N
DFG
3
15
A
N
MT3
5
12
A
N
ATP
6
2
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Chain: A
Legend
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Name
Hit Count
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Chain: A