Co-crystal Structure of PERK bound to N-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1H-pyrazole-4-carboxamide inhibitor

PDB Details

PDB ID
4X7H
Status
CURRENT
Deposition Date
2014-12-09
Modification Date
2015-02-25
Pubmed ID
25587754
Method
X-RAY DIFFRACTION
Resolution (Å)
2.0
UniProt Accessions
Q9NZJ5

Mapping Results

Chain Terminus Site Consensus Site Rank Consensus Site Population
A C DRS 5 9
A C DFG 6 8
A C AAS 7 7
A C PDIG 8 5
A N MT3 0 23
A N MT3 5 5

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Legend

Color Name Hit Count