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Co-crystal Structure of PERK bound to N-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1H-pyrazole-4-carboxamide inhibitor
PDB Details
PDB ID
4X7H
Status
CURRENT
Deposition Date
2014-12-09
Modification Date
2015-02-25
Pubmed ID
25587754
Method
X-RAY DIFFRACTION
Resolution (Å)
2.0
UniProt Accessions
Q9NZJ5
Mapping Results
Chain
Terminus
Site
Consensus Site Rank
Consensus Site Population
A
C
DRS
5
9
A
C
DFG
6
8
A
C
AAS
7
7
A
C
PDIG
8
5
A
N
MT3
0
23
A
N
MT3
5
5
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Chain: A
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Name
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Chain: A